SCHEMBL28170261

SCHEMBL28170261

Cc1cc2cc(C(F)(F)F)ccc2nc1-c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.63
DHODH Q02127 1/20 0.55
DHFR P00374 10/20 0.50
NPBWR1 P48145 1/20 0.49
TOP1 P11387 1/20 0.47
DGAT1 O75907 1/20 0.47
KCNH2 Q12809 1/20 0.47
AKT1 P31749 1/20 0.46
AKT2 P31751 1/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
TYMS P04818 2/20 0.46
BACE1 P56817 1/20 0.45
PTGFR P43088 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31070214 0.80 KDM4E (0.64) DHODHDHFRNPBWR1AKT1AKT2
SCHEMBL28185361 0.79 PDE10A (0.59) PDE10ADHODHKCNH2KDM4EALDH1A1
SCHEMBL28536199 0.79 PDE10A (0.69) PDE10ADHODHKDM4EALDH1A1L3MBTL1
SCHEMBL28529940 0.78 PDE10A (0.73) PDE10ADHODHKDM4EALDH1A1L3MBTL1
SCHEMBL2125225 0.78 PDE10A (1.00) PDE10AKDM4EALDH1A1L3MBTL1
SCHEMBL28170329 0.78 PDE10A (0.58) PDE10ADHODHDHFRKDM4EALDH1A1
SCHEMBL28185368 0.78 PDE10A (0.67) PDE10AKDM4EALDH1A1L3MBTL1PTGFR
SCHEMBL1229501 0.78 KDM4E (0.60) DHODHDHFRNPBWR1AKT1AKT2
SCHEMBL10102671 0.77 DHODH (0.46) DHODHDHFRNPBWR1DGAT1KCNH2
SCHEMBL12352239 0.77 KDM4E (0.69) DHODHDHFRAKT1AKT2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107428691-A Bicyclic formamides of 2 aryl quinoline 4 of substituted N and application thereof 拜耳制药股份公司 2017-12-01 CN disclosed
CN-107074773-A Substituted N, the formamide of 2 biaryl quinolin 4 and application thereof 拜耳制药股份公司 2017-08-18 CN disclosed