SCHEMBL28170451

SCHEMBL28170451

O=C1C=C(c2ccccc2)C(=O)N1Cc1ccc(Cl)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RGS4 P49798 2/20 0.67
ALDH1A1 P00352 5/20 0.51
NPSR1 Q6W5P4 3/20 0.51
MAPT P10636 2/20 0.51
HPGD P15428 2/20 0.51
ALOX12 P18054 2/20 0.51
CACNA1B Q00975 2/20 0.51
APBA1 Q02410 2/20 0.51
LMNA P02545 2/20 0.51
HCRTR1 O43613 1/20 0.51
S1PR4 O95977 1/20 0.51
HSP90AA1 P07900 1/20 0.51
S1PR1 P21453 1/20 0.51
MGLL Q99685 2/20 0.50
FAAH O00519 1/20 0.50
NR1H2 P55055 1/20 0.48
NR1H3 Q13133 1/20 0.48
CES2 O00748 1/20 0.48
BCHE P06276 1/20 0.48
CES1 P23141 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9171007 0.90 RGS4 (0.79) RGS4ALDH1A1NPSR1MAPTHPGD
SCHEMBL28976692 0.86 RGS4 (0.65) RGS4ALDH1A1NPSR1MAPTHPGD
SCHEMBL28976672 0.83 RGS4 (0.65) RGS4ALDH1A1NPSR1MAPTHPGD
SCHEMBL28976684 0.82 RGS4 (0.60) RGS4ALDH1A1NPSR1MAPTHPGD
SCHEMBL2644212 0.82 RGS4 (0.64) RGS4MAPTNR1H2NR1H3GSK3A
SCHEMBL13517162 0.80 RGS4 (1.00) RGS4ALDH1A1NPSR1MAPTHPGD
SCHEMBL28976859 0.79 RGS4 (0.56) RGS4ALDH1A1MAPTLMNATP53
SCHEMBL7861858 0.79 RGS4 (0.59) RGS4ALDH1A1NPSR1MAPTHPGD
SCHEMBL30272716 0.78 RGS4 (0.55) RGS4ALDH1A1MAPTALOX12LMNA
SCHEMBL7774092 0.78 RGS4 (0.58) RGS4ALDH1A1NPSR1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107162950-A N substitution maleimide compounds and its preparation based on pharmaceutical intermediate are studied with antibacterial activity 浙江工业大学 2017-09-15 CN disclosed