SCHEMBL28172736

SCHEMBL28172736

CN(C)C=Cc1cnc(Br)cc1[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.39
BACE1 P56817 2/20 0.35
MAPT P10636 6/20 0.35
ALDH1A1 P00352 4/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ACHE P22303 4/20 0.34
BCHE P06276 2/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
MMP14 P50281 1/20 0.33
RAB9A P51151 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX15 P16050 1/20 0.33
PRKDC P78527 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ERN1 O75460 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19015510 1.00 PTGS2 (0.39) PTGS2BACE1MAPTALDH1A1MAPK1
SCHEMBL29709737 0.88 MAPT (0.35) PTGS2BACE1MAPTALDH1A1MAPK1
SCHEMBL10179458 0.88 MAPT (0.35) PTGS2BACE1MAPTALDH1A1MAPK1
SCHEMBL10179459 0.88 MAPT (0.35) PTGS2BACE1MAPTALDH1A1MAPK1
SCHEMBL406829 0.76 PTGS2 (0.47) PTGS2BACE1MAPTALDH1A1MAPK1
SCHEMBL29996459 0.76 PTGS2 (0.47) PTGS2BACE1MAPTALDH1A1MAPK1
SCHEMBL1096483 0.76 PTGS2 (0.47) PTGS2BACE1MAPTALDH1A1MAPK1
SCHEMBL3133057 0.75 VCP (0.38) PTGS2MAPTALDH1A1MAPK1HTT
SCHEMBL17533407 0.75 CYP1A2 (0.42) PTGS2MAPTALDH1A1MAPK1HTT
SCHEMBL30204572 0.75 VCP (0.38) PTGS2MAPTALDH1A1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104955824-B It is used as the aminopyrimidine compounds of the inhibitor of the EGFR mutant containing T790M 豪夫迈·罗氏有限公司 2017-09-22 CN disclosed