SCHEMBL28175233

SCHEMBL28175233

CS(=O)(=O)CCn1ccc(C2CC2)n1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HCRTR2 O43614 5/20 0.38
RORC P51449 3/20 0.37
KDM1A O60341 1/20 0.35
TLR9 Q9NR96 4/20 0.31
TLR8 Q9NR97 4/20 0.31
TLR7 Q9NYK1 4/20 0.31
JAK2 O60674 2/20 0.31
TYK2 P29597 2/20 0.31
JAK3 P52333 2/20 0.31
JAK1 P23458 1/20 0.31
DDB1 Q16531 1/20 0.30
CRBN Q96SW2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23940711 0.78 NPC1 (0.57) NPC1RAB9ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL2661186 0.75 ALDH1A1 (0.41) ALDH1A1L3MBTL1RORCKDM1A
SCHEMBL21166146 0.74 NPC1 (0.60) NPC1RAB9ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL16877119 0.74 NPC1 (0.56) NPC1RAB9ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL28175220 0.74 NPC1 (0.53) NPC1RAB9ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL16331968 0.73 RORC (0.31) L3MBTL1RORCKDM1A
SCHEMBL28175232 0.72 NPC1 (0.47) NPC1RAB9ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL24015836 0.72 NPC1 (0.47) NPC1RAB9ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL22060805 0.71 NPC1 (0.53) NPC1RAB9ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL17045306 0.71 NPC1 (0.36) NPC1RAB9ASMN1; SMN2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074861-A 9H pyrimido [4,5-B ] indoles and related analogs as BET bromodomain inhibitors 密执安大学评议会 2017-08-18 CN disclosed