SCHEMBL28176103

SCHEMBL28176103

Cc1cc(N)cc(COC(N)=O)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 1/20 0.47
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
TACR1 P25103 11/20 0.40
ALOX15 P16050 1/20 0.39
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
EGFR P00533 1/20 0.36
CACNA1F O60840 1/20 0.36
CACNA1D Q01668 1/20 0.36
CACNA1S Q13698 1/20 0.36
CACNA1C Q13936 1/20 0.36
FFAR1 O14842 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
POLB P06746 1/20 0.36
TOP2A P11388 1/20 0.35
TOP2B Q02880 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL586545 0.93 PARP10 (0.53) PARP10TACR1ALOX15CYP1A2CYP3A4
SCHEMBL11795798 0.78 PARP10 (0.41) PARP10ALDH1A1TACR1ALOX15CYP1A2
SCHEMBL12220491 0.77 NPC1 (0.48) PARP10TACR1CYP1A2CYP3A4EGFR
SCHEMBL7656159 0.75 IDO1 (0.59) FFAR4POLB
SCHEMBL23158847 0.75 ALDH1A1 (0.52) PARP10ALDH1A1TSHRTACR1
SCHEMBL9686081 0.75 ALDH1A1 (0.55) PARP10ALDH1A1TACR1CYP3A4EGFR
SCHEMBL5971176 0.75 ALDH1A1 (0.55) PARP10ALDH1A1TACR1CYP3A4EGFR
SCHEMBL15693295 0.75 ACHE (0.47)
SCHEMBL3297072 0.74 HTT (0.48) ALDH1A1TSHRALOX15POLB
SCHEMBL13586898 0.73 ALDH1A1 (0.53) PARP10ALDH1A1TACR1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107295798-A Benzazepine dicarboxamide compound 豪夫迈·罗氏有限公司 2017-10-24 CN disclosed