SCHEMBL28181583

SCHEMBL28181583

CC1(C)Oc2ccccc2C1Cl

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNE1 P15382 2/20 0.42
KCNQ1 P51787 2/20 0.42
LMNA P02545 2/20 0.35
ABCB1 P08183 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
APOBEC3A P31941 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
HTR2B P41595 1/20 0.33
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HTT P42858 1/20 0.32
CNR1 P21554 1/20 0.32
OPRD1 P41143 1/20 0.32
TSHR P16473 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28240913 0.79 KCNE1 (0.42) KCNE1KCNQ1LMNAABCB1ALDH1A1
SCHEMBL3409162 0.77 KCNE1 (0.38) KCNE1KCNQ1LMNAABCB1ALDH1A1
SCHEMBL28240889 0.77 KCNE1 (0.38) KCNE1KCNQ1LMNAALDH1A1HTR2B
SCHEMBL17929070 0.77 KCNE1 (0.43) KCNE1KCNQ1LMNAABCB1ALDH1A1
SCHEMBL15254619 0.77 KCNE1 (0.43) KCNE1KCNQ1LMNAABCB1ALDH1A1
SCHEMBL28241727 0.76 LMNA (0.35) KCNE1KCNQ1LMNAALDH1A1HTR2B
SCHEMBL24151289 0.75 KCNE1 (0.42) KCNE1KCNQ1LMNAABCB1ALDH1A1
SCHEMBL2818050 0.75 KCNE1 (0.49) KCNE1KCNQ1ABCB1KDM4EMAOA
SCHEMBL28228605 0.75 KCNE1 (0.42) KCNE1KCNQ1LMNAABCB1ALDH1A1
SCHEMBL13380562 0.73 IDO1 (0.44) KCNE1KCNQ1LMNAABCB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108473498-A Pyrazolo [1,5a] pyrimidine derivatives as IRAK4 conditioning agents 豪夫迈·罗氏有限公司 2018-08-31 CN disclosed
CN-105209447-B Bicyclic [2.2.2] sour GPR120 conditioning agents 百时美施贵宝公司 2017-11-21 CN disclosed