SCHEMBL28186295

SCHEMBL28186295

COc1cccc(CN2CC2)c1

nearest known ligand 0.90

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.90
KDM4E B2RXH2 4/20 0.79
ALDH1A1 P00352 4/20 0.79
GAA P10253 1/20 0.73
MEN1 O00255 3/20 0.68
KMT2A Q03164 3/20 0.68
MAPT P10636 1/20 0.67
TSHR P16473 1/20 0.67
HTR1A P08908 1/20 0.66
DRD2 P14416 1/20 0.66
HTR2B P41595 1/20 0.66
CASP1 P29466 1/20 0.64
CASP4 P49662 1/20 0.64
CASP5 P51878 1/20 0.64
ATM Q13315 1/20 0.64
LMNA P02545 1/20 0.63
HTT P42858 1/20 0.63
FAAH O00519 1/20 0.63
TDP1 Q9NUW8 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20804357 1.00 SIGMAR1 (0.90) SIGMAR1KDM4EALDH1A1GAAMEN1
SCHEMBL21733083 0.93 SIGMAR1 (0.79) SIGMAR1KDM4EALDH1A1GAAMEN1
SCHEMBL14076364 0.93 SIGMAR1 (0.79) SIGMAR1KDM4EALDH1A1GAAMEN1
SCHEMBL3162705 0.93 SIGMAR1 (0.79) SIGMAR1KDM4EALDH1A1GAAMEN1
SCHEMBL30774908 0.93 SIGMAR1 (0.79) SIGMAR1KDM4EALDH1A1GAAMEN1
SCHEMBL22642361 0.92 SIGMAR1 (0.77) SIGMAR1KDM4EALDH1A1GAAMEN1
SCHEMBL656952 0.92 SIGMAR1 (0.77) SIGMAR1KDM4EALDH1A1GAAMEN1
SCHEMBL29447356 0.91 SIGMAR1 (0.77) SIGMAR1KDM4EALDH1A1GAAMEN1
SCHEMBL1883482 0.91 SIGMAR1 (0.77) SIGMAR1KDM4EALDH1A1GAAMEN1
SCHEMBL27253620 0.91 SIGMAR1 (0.80) SIGMAR1KDM4EALDH1A1GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107406426-A Cyclic ureas as ROCK inhibitors 百时美施贵宝公司 2017-11-28 CN disclosed