SCHEMBL28186397

SCHEMBL28186397

O=C(O)c1cc(Cl)cc(C[SH](=O)=O)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.57
HCAR1 Q9BXC0 1/20 0.50
HCAR2 Q8TDS4 1/20 0.40
MRGPRX4 Q96LA9 4/20 0.40
TTR P02766 1/20 0.39
RXRA P19793 3/20 0.39
RXRB P28702 3/20 0.39
TSHR P16473 2/20 0.38
ALOX15 P16050 1/20 0.38
YTHDC1 Q96MU7 1/20 0.37
AR P10275 1/20 0.37
RXRG P48443 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NR4A2 P43354 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27966126 0.80 TSHR (0.42) TPMTTSHRALDH1A1
SCHEMBL8979358 0.79 TPMT (0.64) TPMTHCAR1HCAR2MRGPRX4TTR
SCHEMBL28104156 0.78 POLB (0.40) TPMTHCAR2MRGPRX4TTRRXRA
SCHEMBL6954785 0.77 TPMT (0.61) TPMTHCAR1HCAR2MRGPRX4TTR
SCHEMBL27709068 0.76 TPMT (0.59) TPMTHCAR1HCAR2MRGPRX4TTR
SCHEMBL69625 0.75 TPMT (0.89) TPMTHCAR1HCAR2TTRRXRA
SCHEMBL28214359 0.75 TPMT (1.00) TPMTHCAR1HCAR2TTRRXRA
SCHEMBL23699 0.75 TPMT (1.00) TPMTHCAR1HCAR2TTRRXRA
SCHEMBL20494155 0.75 FFAR4 (0.35) MRGPRX4TSHR
SCHEMBL11771738 0.74 TPMT (0.57) TPMTHCAR1HCAR2MRGPRX4TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073748-B New octahydro-pyrrolo- [3,4-c]-azole derivatives as autotaxin inhibitors and the like 豪夫迈·罗氏有限公司 2018-06-01 CN disclosed
CN-104684915-B Novel bicyclic derivative 霍夫曼-拉罗奇有限公司 2017-10-31 CN disclosed