SCHEMBL28189261

SCHEMBL28189261

CC(C)(C)OC(=O)Nc1cccc(Nc2ccnc(Nc3ccccc3)n2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
SYK P43405 4/20 0.56
AURKA O14965 13/20 0.56
CHEK1 O14757 2/20 0.56
PDPK1 O15530 2/20 0.56
CHEK2 O96017 2/20 0.56
PRKCG P05129 2/20 0.56
CDK1 P06493 2/20 0.56
PIM1 P11309 2/20 0.56
FGFR1 P11362 2/20 0.56
FGFR3 P22607 2/20 0.56
RPS6KB1 P23443 2/20 0.56
CDK2 P24941 2/20 0.56
MARK3 P27448 2/20 0.56
MAPK1 P28482 2/20 0.56
EPHA2 P29317 2/20 0.56
BLK P51451 2/20 0.56
RPS6KA3 P51812 2/20 0.56
CSNK2A1 P68400 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30737936 0.88 AURKA (0.56) NPC1RAB9AAURKACHEK1PDPK1
SCHEMBL18780747 0.88 SYK (0.48) NPC1RAB9ASYKAURKAAURKB
SCHEMBL28823474 0.86 SYK (0.52) NPC1RAB9ASYKAURKAAURKB
SCHEMBL28850302 0.84 SYK (0.50) NPC1RAB9ASYKAURKACDK1
SCHEMBL17266536 0.84 JAK3 (0.58) SYKAURKACDK1CDK2IKBKB
SCHEMBL28039312 0.82 SYK (0.48) NPC1RAB9ASYKAURKAAURKB
SCHEMBL28039617 0.81 SYK (0.48) NPC1RAB9ASYKAURKAAURKB
SCHEMBL14769279 0.81 EGFR (0.69) SYKITKEGFRJAK3BTK
SCHEMBL9479889 0.80 MAPT (0.62) RAB9ASYKCDK1MAPK1MAPT
SCHEMBL13921824 0.80 SYK (0.60) SYKMAPK1MAPTITKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727382-A Heterocyclic compound as BTK inhibitor and its application 华东理工大学 2018-11-02 CN disclosed
CN-105985342-B As the pyrimido-pyrimidine derovatives of EGFR inhibitor and its application 华东理工大学 2018-07-24 CN disclosed
CN-107428763-A As the pyrimido-pyrimidine derovatives of EGFR inhibitor and its application 华东理工大学 2017-12-01 CN disclosed