SCHEMBL2819008

SCHEMBL2819008

N#Cc1ccccc1N1CCN(C(=O)[C@@H]2C[C@H](NCCc3cc(C(F)(F)F)cc(C(F)(F)F)c3)CN2Cc2ccccc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 5/20 0.48
TACR1 P25103 1/20 0.40
P2RY12 Q9H244 1/20 0.39
DPP4 P27487 1/20 0.39
NPC1 O15118 1/20 0.39
DRD2 P14416 2/20 0.37
DRD3 P35462 1/20 0.37
CTSL P07711 4/20 0.37
CTSS P25774 4/20 0.37
DRD4 P21917 1/20 0.37
GRM5 P41594 1/20 0.37
CCR2 P41597 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2820849 0.92 CHRM4 (0.47) CHRM4TACR1P2RY12DPP4NPC1
SCHEMBL2817332 0.85 CHRM4 (0.53) CHRM4DRD2DRD3
SCHEMBL2818696 0.84 CHRM4 (0.48) CHRM4P2RY12DPP4NPC1DRD2
SCHEMBL2821338 0.83 DRD2 (0.44) CHRM4DPP4DRD2DRD3CTSL
SCHEMBL13841884 0.83 DRD2 (0.44) CHRM4DPP4DRD2DRD3CTSL
SCHEMBL2818171 0.83 C5AR1 (0.44) CHRM4DPP4DRD2DRD4GRM5
SCHEMBL2819005 0.82 CHRM4 (0.43) CHRM4TACR1DPP4NPC1CTSL
SCHEMBL2821782 0.82 DPP4 (0.45) CHRM4DPP4DRD2DRD3DRD4
SCHEMBL2817206 0.81 CHRM4 (0.42) CHRM4DPP4DRD2DRD4GRM5
SCHEMBL3637803 0.81 CHRM4 (0.42) CHRM4DPP4DRD2DRD4GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155672-B1 PROLINAMIDE DERIVATIVES AS NK3 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-10-27 EP claimed