SCHEMBL28190092

SCHEMBL28190092

COc1cnc(OC)c(N)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.38
CASP1 P29466 1/20 0.38
SIRT6 Q8N6T7 1/20 0.37
AURKA O14965 1/20 0.37
TTK P33981 1/20 0.37
AURKB Q96GD4 1/20 0.37
INCENP Q9NQS7 1/20 0.37
RECQL P46063 2/20 0.35
HTT P42858 1/20 0.35
PIK3CA P42336 3/20 0.34
POLB P06746 2/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33
FGFR1 P11362 2/20 0.33
TDP1 Q9NUW8 1/20 0.32
LMNA P02545 1/20 0.32
NNMT P40261 1/20 0.32
DHFR P00374 1/20 0.31
PIK3CD O00329 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11222657 0.83 SIRT6 (0.37) MAPTCASP1SIRT6AURKATTK
SCHEMBL13114213 0.82 SIRT6 (0.39) SIRT6PIK3CAFGFR1LMNANNMT
SCHEMBL28004405 0.80 SIRT6 (0.41) MAPTSIRT6POLBTDP1NNMT
SCHEMBL11216390 0.80 CDK1 (0.40) MAPTCCNA2CDK2CCNA1
SCHEMBL11217711 0.79 ALDH1A1 (0.44) MAPTCASP1HTTLMNA
SCHEMBL1731975 0.78 HTT (0.39) MAPTCASP1AURKATTKAURKB
SCHEMBL10314188 0.78 SIRT6 (0.37) SIRT6PIK3CAFGFR1LMNANNMT
SCHEMBL29395867 0.78 HTT (0.39) MAPTCASP1AURKATTKAURKB
SCHEMBL1731368 0.77 CCR4 (0.38) MAPTCASP1AURKATTKAURKB
SCHEMBL1315972 0.77 SIRT6 (0.36) SIRT6HTTPIK3CAFGFR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107519168-A A kind of application of NRF2 inhibitor and its related compound treatment tuberculosis infection 中国医科大学 2017-12-29 CN disclosed