SCHEMBL28197850

SCHEMBL28197850

NNOC(=O)c1ccc(C(=O)O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.52
TP53 P04637 1/20 0.52
ALDH1A1 P00352 3/20 0.48
MAPT P10636 3/20 0.48
POLB P06746 1/20 0.48
KMT2A Q03164 1/20 0.48
SRD5A2 P31213 2/20 0.46
CA1 P00915 5/20 0.44
CA2 P00918 5/20 0.44
CA12 O43570 3/20 0.44
CA9 Q16790 3/20 0.44
CA3 P07451 2/20 0.44
CA6 P23280 2/20 0.44
CA5A P35218 2/20 0.44
CA7 P43166 2/20 0.44
CA14 Q9ULX7 2/20 0.44
CA5B Q9Y2D0 2/20 0.44
TYR P14679 1/20 0.44
DRD1 P21728 1/20 0.44
CA4 P22748 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9551766 0.98 TSHR (0.50) TSHRTP53ALDH1A1MAPTPOLB
SCHEMBL9847967 0.91 MAPT (0.50) TSHRALDH1A1MAPTPOLBKMT2A
SCHEMBL3035584 0.84 ALDH1A1 (0.67) TSHRTP53ALDH1A1MAPTPOLB
SCHEMBL7051844 0.83 CA12 (0.59) TSHRALDH1A1MAPTPOLBKMT2A
SCHEMBL1002998 0.81 KMT2A (0.42) ALDH1A1MAPTPOLBKMT2ACA1
SCHEMBL8167020 0.81 ALDH1A1 (0.59) TSHRTP53ALDH1A1MAPTPOLB
SCHEMBL11856189 0.78 TSHR (0.52) TSHRTP53ALDH1A1MAPTPOLB
SCHEMBL17510000 0.78 CA1 (0.68) TP53ALDH1A1MAPTKMT2ACA1
SCHEMBL3908499 0.77 CYP1A2 (0.55) TSHRALDH1A1MAPTPOLBKMT2A
SCHEMBL7219677 0.75 TSHR (0.60) TSHRTP53ALDH1A1SRD5A2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108883196-A Target the antibody-drug conjugates of GCC 米伦纽姆医药公司 2018-11-23 CN disclosed
CN-108290895-A Process for preparing cytotoxic benzodiazepine derivatives 伊缪诺金公司 2018-07-17 CN disclosed
CN-107708810-A Conjugates of cysteine engineered antibodies 伊缪诺金公司 2018-02-16 CN disclosed
CN-107580604-A Conjugate comprising cell binding agent and cytotoxic agent 伊缪诺金公司 2018-01-12 CN disclosed