Pentostatin

Pentostatin

SCHEMBL28197957

CNNCc1ccc(C(=O)NC(C)C)cc1.OC[C@H]1O[C@@H](n2cnc3c2NC=NC[C@H]3O)C[C@@H]1O

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADA

The experimentally established mechanism targets of Pentostatin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADA known ✓ P00813 3/20 0.63
ADORA3 P0DMS8 1/20 0.63
ADORA2A P29274 1/20 0.63
ADORA1 P30542 1/20 0.63
AMPD3 Q01432 4/20 0.45
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
PTGS2 P35354 1/20 0.43
AMPD2 Q01433 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pentostatin SCHEMBL2045053 0.79 ADA (1.00) ADAADORA3ADORA2AADORA1AMPD3
Pentostatin SCHEMBL14031902 0.79 ADA (1.00) ADAADORA3ADORA2AADORA1AMPD3
Pentostatin SCHEMBL1649740 0.79 ADA (1.00) ADAADORA3ADORA2AADORA1AMPD3
Pentostatin SCHEMBL2818 0.79 ADA (1.00) ADAADORA3ADORA2AADORA1AMPD3
Pentostatin SCHEMBL28886873 0.77 ADA (0.90) ADAADORA3ADORA2AADORA1AMPD3
Pentostatin SCHEMBL28078896 0.71 ADA (0.77) ADAADORA3ADORA2AADORA1AMPD3
Promethazine SCHEMBL28095270 0.70 ADA (0.65) ADAADORA3ADORA2AADORA1AMPD3
Pentostatin SCHEMBL28265748 0.68 ADA (0.64) ADAADORA3ADORA2AADORA1AMPD3
Procarbazine SCHEMBL2304032 0.64 ALDH1A1 (0.97) ALDH1A1LMNACYP1A2ALOX15CYP2C19
Procarbazine SCHEMBL29196982 0.64 ALDH1A1 (0.97) ALDH1A1LMNACYP1A2ALOX15CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108700590-A Cell population analysis 英国质谱公司 2018-10-23 CN disclosed
CN-107667288-A Spectral analysis of microorganisms 英国质谱公司 2018-02-06 CN disclosed