SCHEMBL2819819

SCHEMBL2819819

COCCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc(N4CCCC4=O)cc3)NC(=O)O)C2)c(C)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 2/20 0.41
CNR2 P34972 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PSMB5 P28074 1/20 0.35
CTSD P07339 8/20 0.35
BACE1 P56817 8/20 0.35
BACE2 Q9Y5Z0 8/20 0.35
METTL3 Q86U44 1/20 0.34
METTL14 Q9HCE5 1/20 0.34
TSHR P16473 1/20 0.34
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
ACACB O00763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7903380 0.92 PROKR1 (0.39) PROKR1CNR2PSMB5TSHR
SCHEMBL2790786 0.90 PROKR1 (0.44) PROKR1CNR2CYP1A2MEN1KMT2A
SCHEMBL2790497 0.90 PROKR1 (0.45) PROKR1CNR2KMT2ATSHRALDH1A1
SCHEMBL2789452 0.90 PROKR1 (0.45) PROKR1CNR2KMT2ATSHRALDH1A1
SCHEMBL2789222 0.88 PROKR1 (0.41) PROKR1CNR2CYP1A2CYP2D6CYP2C9
SCHEMBL742501 0.87 MAPT (0.43) CYP2D6ALDH1A1
SCHEMBL742502 0.87 MAPT (0.43) CYP2D6ALDH1A1
SCHEMBL2877866 0.85 PROKR1 (0.40) PROKR1CNR2CYP1A2MEN1KMT2A
SCHEMBL2789132 0.84 PROKR1 (0.38) PROKR1CNR2MEN1KMT2A
SCHEMBL2788887 0.83 PROKR1 (0.39) PROKR1CNR2KMT2ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed