SCHEMBL28200955

SCHEMBL28200955

CC(NC(=O)OC(C)(C)C)c1cc[nH]c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.43
KMT2A Q03164 2/20 0.41
TSHR P16473 2/20 0.40
HSD17B10 Q99714 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CTSS P25774 1/20 0.39
ATM Q13315 2/20 0.38
MAPT P10636 1/20 0.38
TRPA1 O75762 1/20 0.38
MEN1 O00255 1/20 0.37
ABCB1 P08183 1/20 0.37
CA4 P22748 1/20 0.36
CA9 Q16790 1/20 0.36
EPHX2 P34913 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28200954 1.00 CTSK (0.43) CTSKKMT2ATSHRHSD17B10CA1
SCHEMBL27509373 0.78 ATM (0.54) CTSKKMT2ATSHRHSD17B10CTSS
SCHEMBL12203593 0.78 CTSK (0.62) CTSKKMT2AHSD17B10CTSSATM
SCHEMBL6346032 0.78 CTSK (0.62) CTSKKMT2AHSD17B10CTSSATM
SCHEMBL6346030 0.78 CTSK (0.62) CTSKKMT2AHSD17B10CTSSATM
SCHEMBL23205455 0.76 GPR139 (0.48) CTSKKMT2ATSHRHSD17B10CA1
SCHEMBL13542547 0.76 GPR139 (0.48) CTSKKMT2ATSHRHSD17B10CA1
SCHEMBL3502878 0.76 CTSK (0.48) CTSKKMT2ATSHRHSD17B10CA1
SCHEMBL15048272 0.76 CTSK (0.48) CTSKKMT2ATSHRHSD17B10CA1
SCHEMBL25546987 0.76 GPR139 (0.48) CTSKKMT2ATSHRHSD17B10CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105263935-B 6, 7-dihydropyrazolo [1,5-a ] pyrazin-4 (5H) -one compounds and their use as negative allosteric modulators of the MG L UR2 receptor 詹森药业有限公司 2018-02-27 CN disclosed