SCHEMBL28201449

SCHEMBL28201449

c1ccc(Cc2nc3cc(-c4ccccc4)ccc3s2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.49
LIPG Q9Y5X9 8/20 0.44
KDM4E B2RXH2 2/20 0.43
PIK3CA P42336 2/20 0.43
PI4KA P42356 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
PIK3CD O00329 1/20 0.42
PIK3CB P42338 1/20 0.42
PIK3CG P48736 1/20 0.42
NPC1 O15118 1/20 0.42
HPGD P15428 1/20 0.42
NFKB1 P19838 1/20 0.42
STAT1 P42224 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28201976 0.88 LOXL2 (0.46) HDAC6LIPG
SCHEMBL203384 0.83 PIK3CA (0.44) HDAC6LIPGKDM4EPIK3CAPI4KA
SCHEMBL2956510 0.81 LOXL2 (0.62) HDAC6NPC1HPGDRAB9AMEN1
SCHEMBL5074923 0.81 AKR1B1 (0.46) HDAC6KDM4ENPC1RAB9AMEN1
SCHEMBL3190308 0.81 KDM4E (0.51) HDAC6KDM4ENPC1HPGDNFKB1
SCHEMBL28984547 0.81 MAPT (0.47) HDAC6KDM4ENPC1RAB9AMEN1
SCHEMBL28984552 0.81 HDAC6 (0.55) HDAC6KDM4ENPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL3898824 0.80 KDM4E (0.50) HDAC6KDM4ENPC1HPGDNFKB1
SCHEMBL1127709 0.80 UBE2T (0.61) KDM4ENPC1HPGDRAB9AMEN1
SCHEMBL12596792 0.78 PIK3CA (0.58) LIPGKDM4EPIK3CAPI4KAPI4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103214471-B The preparation method of compound with Na-dependent glucose transporter inhibitory activity 田边三菱制药株式会社 2018-02-06 CN disclosed