SCHEMBL28201461

SCHEMBL28201461

COc1c(Cc2cc3ccccc3s2)c(Br)cc2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.44
AGXT P21549 1/20 0.44
ADRB2 P07550 1/20 0.44
ASIC3 Q9UHC3 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
TUBB4A P04350 4/20 0.39
TUBB P07437 4/20 0.39
TUBA3C P0DPH7 4/20 0.39
TUBA1B P68363 4/20 0.39
TUBA4A P68366 4/20 0.39
TUBB4B P68371 4/20 0.39
TUBB3 Q13509 4/20 0.39
TUBB2A Q13885 4/20 0.39
TUBB8 Q3ZCM7 4/20 0.39
TUBA3E Q6PEY2 4/20 0.39
TUBA1A Q71U36 4/20 0.39
TUBA1C Q9BQE3 4/20 0.39
TUBB6 Q9BUF5 4/20 0.39
TUBB2B Q9BVA1 4/20 0.39
TUBB1 Q9H4B7 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1775820 0.80 CYP2A6 (0.44) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL155195 0.77 CYP2A6 (0.42) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL28954990 0.76 CYP2A6 (0.47) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL1773869 0.72 CYP2A6 (0.47) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL16018691 0.72 CYP2A6 (0.42) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL6958014 0.71 TUBB4A (0.53) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL1539306 0.71 SLC5A2 (0.55) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL12425721 0.71 SLC5A2 (0.50) CYP2A6AGXTADRB2ASIC3LOXL2
SCHEMBL29227832 0.70 ALDH1A1 (0.48) CYP2A6TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL4961407 0.70 CYP2A6 (0.69) CYP2A6AGXTADRB2ASIC3LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103214471-B The preparation method of compound with Na-dependent glucose transporter inhibitory activity 田边三菱制药株式会社 2018-02-06 CN disclosed