SCHEMBL28205337

SCHEMBL28205337

COC(=O)c1cnc(Cl)cn1.[NaH]

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 2/20 0.55
MAPK1 P28482 4/20 0.50
KDM4E B2RXH2 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
JUN P05412 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
PCSK9 Q8NBP7 1/20 0.42
LCK P06239 1/20 0.41
GABRP O00591 2/20 0.39
GABRD O14764 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GABRA1 P14867 2/20 0.39
GABRB1 P18505 2/20 0.39
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRA5 P31644 2/20 0.39
GABRA3 P34903 2/20 0.39
GABRA2 P47869 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL64740 0.98 SIRT6 (0.57) SIRT6MAPK1KDM4EL3MBTL1JUN
SCHEMBL30196970 0.98 SIRT6 (0.57) SIRT6MAPK1KDM4EL3MBTL1JUN
SCHEMBL68869 0.85 MAPK1 (0.63) SIRT6MAPK1KDM4EL3MBTL1PCSK9
SCHEMBL2646157 0.78 SIRT6 (0.52) SIRT6JUNNFKB1NFKB2RELA
SCHEMBL30986210 0.78 SIRT6 (0.52) SIRT6MAPK1KDM4EL3MBTL1GABRP
SCHEMBL31515460 0.78 SIRT6 (0.52) SIRT6JUNNFKB1NFKB2RELA
SCHEMBL7999648 0.78 SIRT6 (0.52) SIRT6MAPK1KDM4EL3MBTL1GABRP
SCHEMBL990711 0.78 MAPK1 (0.55) SIRT6MAPK1KDM4EL3MBTL1PCSK9
SCHEMBL5700876 0.78 KDM4E (0.61) SIRT6MAPK1KDM4EL3MBTL1PCSK9
SCHEMBL25153862 0.76 MAPK1 (0.46) MAPK1KDM4EL3MBTL1LCKGABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849056-A BACE1 inhibitor 2 amino 7A phenyl 3,4,4A, 5,7,7A hexahydro furyl simultaneously [3,4 B] pyridine H.隆德贝克有限公司 2018-03-27 CN disclosed