SCHEMBL28211519

SCHEMBL28211519

CNC(=O)Cc1cccc(CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GLS O94925 16/20 0.62
BRD4 O60885 2/20 0.45
KDM4A O75164 1/20 0.45
CREBBP Q92793 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2787151 0.86 GLS (0.58) GLSBRD4KDM4ACREBBP
SCHEMBL13853709 0.86 GLS (0.53) GLSBRD4KDM4ACREBBPCYP3A4
SCHEMBL16181822 0.86 GLS (0.55) GLSBRD4KDM4ACREBBPCYP3A4
SCHEMBL14986954 0.85 GLS (0.57) GLSBRD4KDM4ACREBBP
SCHEMBL8786913 0.85 GLS (0.57) GLSBRD4KDM4ACREBBP
SCHEMBL27113182 0.84 GLS (0.54) GLSBRD4KDM4ACREBBPCYP3A4
SCHEMBL15782622 0.84 GLS (0.69) GLSBRD4KDM4ACREBBP
SCHEMBL13981921 0.83 GLS (0.55) GLSBRD4KDM4ACREBBPCYP3A4
SCHEMBL30069429 0.83 GLS (0.55) GLSBRD4KDM4ACREBBPCYP3A4
SCHEMBL8342682 0.83 GLS (0.55) GLSBRD4KDM4ACREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849044-A Thriazaspiro last of the ten Heavenly stems ketone compounds as DDR1 inhibitor 豪夫迈·罗氏有限公司 2018-03-27 CN disclosed