SCHEMBL28212946

SCHEMBL28212946

Cc1cccc(Nc2cc(N)ccn2)c1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 3/20 0.54
EGFR P00533 9/20 0.52
ERBB2 P04626 1/20 0.52
KARS1 Q15046 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49
KCNH2 Q12809 1/20 0.48
SCN5A Q14524 1/20 0.48
SCN9A Q15858 1/20 0.48
KMT2A Q03164 1/20 0.46
ABL1 P00519 1/20 0.46
ABL2 P42684 1/20 0.46
GRM4 Q14833 1/20 0.46
RAB9A P51151 1/20 0.46
RAPGEF4 Q8WZA2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18772775 0.86 TNNI3K (0.59) TNNI3KEGFRKARS1NPSR1KMT2A
SCHEMBL690632 0.83 EGFR (0.62) TNNI3KEGFRERBB2KMT2AABL1
SCHEMBL30216764 0.81 KCNH2 (0.58) EGFRKCNH2SCN5ASCN9AKMT2A
SCHEMBL23588551 0.81 KCNH2 (0.58) EGFRKCNH2SCN5ASCN9AKMT2A
SCHEMBL13166084 0.80 TNNI3K (0.63) TNNI3KEGFRABL1RAB9A
SCHEMBL29645155 0.79 ROCK1 (0.68) TNNI3KEGFR
SCHEMBL8798667 0.79 EGFR (0.61) TNNI3KEGFRERBB2NPSR1ABL1
SCHEMBL6837492 0.78 RAB9A (0.63) TNNI3KEGFRNPSR1KMT2AGRM4
SCHEMBL1387302 0.78 EGFR (0.72) TNNI3KEGFRERBB2NPSR1KMT2A
SCHEMBL5575226 0.77 MAPT (0.67) EGFRERBB2NPSR1KMT2AABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922387-A HETEROCYCLIC INHIBITORS OF ERK1 AND ERK2 AND THEIR USE IN THE TREATMENT OF CANCER 阿沙纳生物科学公司 2018-04-17 CN disclosed