SCHEMBL28215196

SCHEMBL28215196

C[C](C)CN1CCC(CCOCc2ccccc2Br)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 1/20 0.43
PRMT6 Q96LA8 1/20 0.43
ATM Q13315 1/20 0.42
HRH3 Q9Y5N1 2/20 0.39
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
FAAH O00519 1/20 0.38
CHRM3 P20309 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
RECQL P46063 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
DRD2 P14416 1/20 0.37
KDM4E B2RXH2 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HTR1A P08908 1/20 0.36
SLC6A4 P31645 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15845807 0.83 CARM1 (0.44) CARM1PRMT6ATMHRH3HTR2A
SCHEMBL15845660 0.81 ATM (0.43) CARM1PRMT6ATMHRH3HTR2A
SCHEMBL15845586 0.79 TEAD1 (0.44) ATMSIGMAR1FAAHCHRM3ALDH1A1
SCHEMBL28036593 0.78 FAAH (0.36) CARM1PRMT6ATMSIGMAR1FAAH
SCHEMBL15845815 0.77 KDM4E (0.51) KDM4E
SCHEMBL15845824 0.75 IDO1 (0.41) CHRM3SLC6A4
SCHEMBL18171754 0.68 IDO1 (0.57) CARM1PRMT6CHRM3ALDH1A1TSHR
SCHEMBL18171753 0.68 IDO1 (0.57) CARM1PRMT6CHRM3ALDH1A1TSHR
Tert-Butyl Formate SCHEMBL28036594 0.68 SLC6A4 (0.35) CHRM3ALDH1A1SLC6A4
SCHEMBL18171748 0.68 IDO1 (0.61) CARM1PRMT6CHRM3ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903300-B COMT inhibitor 霍夫曼-拉罗奇有限公司 2018-04-17 CN disclosed