SCHEMBL28036593

SCHEMBL28036593

CC(C)(C)C(=O)ON1CCC(CCOCc2ccccc2Br)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.36
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
CHRM3 P20309 2/20 0.35
ATM Q13315 1/20 0.35
MAPT P10636 2/20 0.35
RAB9A P51151 2/20 0.35
PKM P14618 2/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
TEAD1 P28347 1/20 0.34
TEAD3 Q99594 1/20 0.34
SSTR1 P30872 2/20 0.34
SSTR4 P31391 2/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 3/20 0.33
SIGMAR1 Q99720 1/20 0.33
RIPK1 Q13546 1/20 0.33
NPC1 O15118 1/20 0.33
PARP10 Q53GL7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27659695 0.83 AGTR2 (0.44) CHRM3KMT2ATEAD3ALDH1A1SIGMAR1
SCHEMBL15845815 0.83 KDM4E (0.51) PKMKDM4E
SCHEMBL28772120 0.82 GPR119 (0.39) CHRM3RIPK1
SCHEMBL15845586 0.81 TEAD1 (0.44) FAAHCHRM3ATMMAPTRAB9A
SCHEMBL15845807 0.80 CARM1 (0.44) CARM1PRMT6CHRM3ATMSSTR1
SCHEMBL28215196 0.78 CARM1 (0.43) FAAHCARM1PRMT6CHRM3ATM
SCHEMBL28227977 0.76 LMNA (0.46) CARM1PRMT6CHRM3RAB9APKM
SCHEMBL27897795 0.76 ADAM17 (0.34) FAAH
SCHEMBL27719651 0.74 ALDH1A1 (0.39) RAB9AALDH1A1KDM4ESIGMAR1
SCHEMBL15845660 0.74 ATM (0.43) FAAHCARM1PRMT6ATMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903300-A Comt inhibitors HOFFMANN LA ROCHE 2015-09-09 CN disclosed