SCHEMBL28215481

SCHEMBL28215481

O=C(O)c1cc(Cc2ccc(OC(F)F)cc2)cc(C(=O)O)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.58
PPARG P37231 3/20 0.48
PPARA Q07869 3/20 0.48
SRD5A2 P31213 1/20 0.47
ATM Q13315 1/20 0.47
ALKBH1 Q13686 1/20 0.45
ALOX15 P16050 1/20 0.45
GFER P55789 1/20 0.45
ADAM17 P78536 1/20 0.45
LMNA P02545 3/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 3/20 0.43
TSHR P16473 1/20 0.43
PTGER4 P35408 1/20 0.42
NLRP3 Q96P20 1/20 0.42
KMT2A Q03164 2/20 0.41
CPT1A P50416 1/20 0.41
CPT1B Q92523 1/20 0.41
HTT P42858 2/20 0.41
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1018588 0.77 KMT2A (0.64) MRGPRX4SRD5A2ATMALOX15GFER
SCHEMBL27893362 0.77 MRGPRX4 (0.47) MRGPRX4ATMALOX15GFERADAM17
SCHEMBL28951143 0.77 SRD5A2 (0.58) SRD5A2LMNAPOLBMAPTTSHR
SCHEMBL28029673 0.76 PPARA (0.49) MRGPRX4PPARASRD5A2LMNAKMT2A
SCHEMBL28247826 0.76 PPARG (0.59) MRGPRX4PPARGPPARAALOX15LMNA
Hydrochloric Acid SCHEMBL9015381 0.76 KMT2A (0.62) MRGPRX4SRD5A2ATMALOX15GFER
SCHEMBL1950244 0.75 CA12 (0.48) SRD5A2ALOX15LMNAMAPTTSHR
SCHEMBL7945362 0.74 ESR1 (0.56) SRD5A2KMT2AMEN1
SCHEMBL4235825 0.74 MRGPRX4 (0.47) MRGPRX4ATMALOX15GFERADAM17
SCHEMBL2142442 0.74 PLA2G10 (0.53) SRD5A2LMNATSHRKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107903251-A Pyrazole formylamine derivate as the TAAR conditioning agents for treating several conditions such as depression, diabetes and Parkinson's 霍夫曼-拉罗奇有限公司 2018-04-13 CN disclosed