SCHEMBL28215694

SCHEMBL28215694

COc1ccc(-c2ncnc(-c3ccc(Cl)cc3)n2)c(OC(C)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.50
HPGD P15428 3/20 0.43
ALDH1A1 P00352 1/20 0.43
F2 P00734 1/20 0.43
GLA P06280 1/20 0.43
POLB P06746 1/20 0.43
NPSR1 Q6W5P4 2/20 0.43
KMT2A Q03164 6/20 0.43
MAPT P10636 4/20 0.43
MEN1 O00255 5/20 0.42
ADORA3 P0DMS8 1/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
AMY1A P0DUB6 1/20 0.40
LMNA P02545 1/20 0.40
DHODH Q02127 1/20 0.39
CYP17A1 P05093 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
NPC1 O15118 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28215172 0.93 BACE1 (0.58) BACE1HPGDALDH1A1F2GLA
SCHEMBL19490331 0.79 ADORA3 (0.60) BACE1HPGDALDH1A1F2GLA
SCHEMBL8383100 0.73 SIRT2 (0.46) POLBNPSR1KMT2AMAPTMEN1
SCHEMBL28809220 0.72 KMT2A (0.43) POLBNPSR1KMT2AMAPTMEN1
SCHEMBL7771404 0.71 NPC1 (0.55) ALDH1A1KMT2AMAPTMEN1ADORA3
SCHEMBL28849727 0.69 CLK4 (0.61) ALDH1A1NPSR1KMT2AMAPTMEN1
SCHEMBL28389589 0.69 MAPT (0.54) KMT2AMAPTMEN1LMNANPC1
SCHEMBL28247350 0.69 NCOA1 (0.56) BACE1HPGDALDH1A1NPSR1KMT2A
SCHEMBL4644027 0.68 BACE1 (0.56) BACE1HPGDALDH1A1F2GLA
SCHEMBL12228435 0.68 KMT2A (0.50) HPGDNPSR1KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108069916-A A kind of 2,4- diaryl for preparing phenyl ring ortho position acetoxylation substitutes the method for -1,3,5 pyrrolotriazine derivatives 中国科学院大连化学物理研究所 2018-05-25 CN disclosed