SCHEMBL28217604

SCHEMBL28217604

NC(=O)N(c1ccccc1)c1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.44
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
KDR P35968 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
S1PR1 P21453 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
MEN1 O00255 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4246399 0.93 HTR3E (0.49) GRM4HTR3EHTR3BHTR3AHTR3D
SCHEMBL1525499 0.90 HTR3E (0.44) GRM4HTR3EHTR3BHTR3AHTR3D
SCHEMBL30019653 0.90 HTR3E (0.44) GRM4HTR3EHTR3BHTR3AHTR3D
SCHEMBL1513968 0.89 NPFFR2 (0.43) GRM4HTR3EHTR3BHTR3AHTR3D
SCHEMBL27734542 0.89 HTR3E (0.43) GRM4HTR3EHTR3BHTR3AHTR3D
SCHEMBL1513809 0.89 HTR3E (0.43) GRM4HTR3EHTR3BHTR3AHTR3D
SCHEMBL58712 0.88 GRM4 (0.46) GRM4KDRLMNASMN1; SMN2USP2
SCHEMBL27514280 0.88 TRPV1 (0.43) GRM4HTR3EHTR3BHTR3AHTR3D
SCHEMBL28217568 0.85 GRM4 (0.43) GRM4ALDH1A1NPSR1POLQ
SCHEMBL27907319 0.83 S1PR1 (0.39) GRM4HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026035-A Compounds having protein tyrosine phosphatase SHP-1 agonist activity 陈昆锋 2018-05-11 CN disclosed