SCHEMBL28218802

SCHEMBL28218802

NNC(=O)c1ccc(C[CH]CCc2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.53
HDAC8 Q9BY41 3/20 0.50
ALDH1A1 P00352 2/20 0.50
MAPT P10636 2/20 0.50
CYP2D6 P10635 1/20 0.46
HDAC6 Q9UBN7 3/20 0.44
HDAC2 Q92769 1/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
MPO P05164 1/20 0.43
CYP3A4 P08684 1/20 0.43
KDM5A P29375 1/20 0.43
BLM P54132 1/20 0.43
GFER P55789 1/20 0.43
PMP22 Q01453 1/20 0.43
HIF1A Q16665 1/20 0.43
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9702631 0.84 GPR52 (0.47) HDAC1HDAC8ALDH1A1HTTGPR52
SCHEMBL28583909 0.84 HDAC1 (0.72) HDAC1HDAC8ALDH1A1MAPTCYP2D6
SCHEMBL364290 0.78 MAOB (0.52) ALDH1A1SMN1; SMN2GPR52
SCHEMBL5471298 0.77 PLA2G10 (0.66) HDAC1HDAC8ALDH1A1MAPTHDAC6
SCHEMBL9219296 0.75 ESR1 (0.48) ALDH1A1KDM4E
SCHEMBL31454334 0.74 HDAC6 (0.74) HDAC1HDAC8ALDH1A1MAPTHDAC6
SCHEMBL10582013 0.72 TSHR (0.47) ALDH1A1MAPTCYP2D6NPC1CYP3A4
Benzoic Acid Hydrazide SCHEMBL83514 0.72 CYP3A4 (0.62) HDAC1HDAC8ALDH1A1MAPTCYP2D6
Benzoic Acid Hydrazide SCHEMBL4515671 0.72 CYP3A4 (0.62) HDAC1HDAC8ALDH1A1MAPTCYP2D6
SCHEMBL20078583 0.72 CYP3A4 (0.62) HDAC1HDAC8ALDH1A1MAPTCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137518-A As 6 inhibitor of histone deacetylase 1,3,4- oxadiazole derivatives compound and include its pharmaceutical composition 株式会社钟根堂 2018-06-08 CN disclosed