SCHEMBL28219902

SCHEMBL28219902

FC(F)(F)CCCOc1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 7/20 0.56
CHRNA4 P43681 7/20 0.56
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP19A1 P11511 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.43
CHRNA3 P32297 2/20 0.43
CHRNA7 P36544 2/20 0.43
MAOB P27338 1/20 0.43
CHRNA1 P02708 1/20 0.43
CHRNG P07510 1/20 0.43
CHRNB1 P11230 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRND Q07001 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28028484 0.91 CHRNB2 (0.60) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL6750074 0.80 CHRNB2 (0.51) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL29656789 0.80 CHRNB2 (0.51) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL1875084 0.78 CHRNB2 (0.62) CHRNB2CHRNA4CYP3A4CYP2D6CYP19A1
SCHEMBL28265183 0.78 MAOB (0.44) MAOB
SCHEMBL30461625 0.78 CHRNB2 (0.62) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL19875367 0.78 CHRNB2 (0.62) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL28193581 0.77 KCNA3 (0.62) MAOB
SCHEMBL12667879 0.77 CHRNB2 (0.62) CHRNB2CHRNA4CYP3A4CYP2D6CYP19A1
SCHEMBL4490294 0.77 CHRNB2 (0.61) CHRNB2CHRNA4CYP3A4CYP2D6CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137579-A Bridging piperidine derivative 豪夫迈·罗氏有限公司 2018-06-08 CN disclosed