SCHEMBL28219972

SCHEMBL28219972

Cc1nc2cccc(Cl)c2c(F)c1Cl

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.46
ELANE P08246 3/20 0.39
PDE2A O00408 2/20 0.39
PDE10A Q9Y233 2/20 0.39
PBRM1 Q86U86 2/20 0.38
DHODH Q02127 1/20 0.38
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
ACHE P22303 2/20 0.36
BCHE P06276 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL537851 0.86 PARP1 (0.46) PARP1ELANEPDE2APDE10AACHE
SCHEMBL4787075 0.79 PARP1 (0.46) PARP1ELANEPDE2APDE10APBRM1
SCHEMBL538143 0.76 PARP1 (0.42) PARP1ELANEPBRM1GRIN1GRIN2A
SCHEMBL27810585 0.74 GPR3 (0.53) PDE10A
SCHEMBL28311772 0.73 GPR3 (0.57) PARP1ELANEPDE2APDE10APBRM1
SCHEMBL12501261 0.72 PARP1 (0.50) PARP1ELANEPBRM1DHODHGRIN1
SCHEMBL29008939 0.71 PARP1 (0.46) PARP1ELANEPBRM1DHODHGRIN1
SCHEMBL4748400 0.69 MAPT (0.52) PARP1ELANEPBRM1DHODHGRIN1
SCHEMBL12501259 0.69 PARP1 (0.47) PARP1ELANEPBRM1DHODHGRIN1
SCHEMBL7417855 0.68 PARP1 (0.50) PARP1ELANEPBRM1DHODHGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137547-A It can be used as the heterocyclic compound of TNF α conditioning agent 百时美施贵宝公司 2018-06-08 CN disclosed