SCHEMBL4787075

SCHEMBL4787075

Cc1nc2cccc(Cl)c2c(O)c1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.46
DHODH Q02127 2/20 0.40
ELANE P08246 2/20 0.39
PBRM1 Q86U86 2/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
STAT3 P40763 1/20 0.38
PDE2A O00408 1/20 0.38
PDE10A Q9Y233 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
TSHR P16473 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28219972 0.79 PARP1 (0.46) PARP1DHODHELANEPBRM1PDE2A
SCHEMBL28219983 0.79 TSHR (0.40) PARP1DHODHELANEKDM4EALDH1A1
SCHEMBL626362 0.75 DYRK1A (0.49) PARP1DHODHELANEKDM4EALDH1A1
Water SCHEMBL25347465 0.73 DYRK1A (0.48) PARP1DHODHELANEKDM4EALDH1A1
SCHEMBL29344431 0.73 PARP1 (0.47) PARP1DHODHELANEPBRM1KDM4E
SCHEMBL28311772 0.73 GPR3 (0.57) PARP1DHODHELANEPBRM1ALDH1A1
SCHEMBL12501261 0.72 PARP1 (0.50) PARP1DHODHELANEPBRM1KDM4E
SCHEMBL29008939 0.71 PARP1 (0.46) PARP1DHODHELANEPBRM1GRIN1
SCHEMBL4788222 0.71 PARP1 (0.46) PARP1DHODHELANEPBRM1KDM4E
SCHEMBL18488814 0.70 CYP1A2 (0.36) KDM4EALDH1A1MEN1KMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117079-A1 ANTIMICROBIAL COMPOUNDS BASED UPON 4-AMINOQUINOLINE HELPERBY THERAPEUTICS LIMITED (GB) 2008-10-02 WO disclosed