SCHEMBL28219987

SCHEMBL28219987

Oc1cc(Br)nc2cccc(Cl)c12

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GLA P06280 1/20 0.42
NQO2 P16083 2/20 0.42
ELANE P08246 2/20 0.39
PARP1 P09874 1/20 0.39
CSNK2A2 P19784 2/20 0.37
CSNK2B P67870 2/20 0.37
CSNK2A1 P68400 2/20 0.37
GRIN1 Q05586 3/20 0.36
GRIN2A Q12879 3/20 0.36
ACHE P22303 3/20 0.36
TSHR P16473 1/20 0.36
BCHE P06276 1/20 0.36
DHFR P00374 1/20 0.36
PBRM1 Q86U86 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26607337 0.85 PARP1 (0.43) ELANEPARP1GRIN1GRIN2AACHE
SCHEMBL8127676 0.81 NQO2 (0.44) KDM4EALDH1A1GLANQO2ELANE
SCHEMBL4788222 0.79 PARP1 (0.46) KDM4EALDH1A1GLANQO2ELANE
SCHEMBL7524860 0.75 KDM4E (0.44) KDM4EALDH1A1NQO2PARP1TSHR
SCHEMBL10611217 0.75 SMN1; SMN2 (0.46) KDM4EALDH1A1GLAACHE
SCHEMBL11828023 0.75 NT5E (0.43) KDM4EALDH1A1GLANQO2ELANE
SCHEMBL9398456 0.73 GRM2 (0.46) NQO2PARP1
SCHEMBL28219983 0.71 TSHR (0.40) KDM4EALDH1A1NQO2ELANEPARP1
SCHEMBL9397215 0.71 PARP1 (0.37) KDM4EALDH1A1GLANQO2ELANE
SCHEMBL9379118 0.70 NQO2 (0.51) KDM4EALDH1A1NQO2PARP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137547-A It can be used as the heterocyclic compound of TNF α conditioning agent 百时美施贵宝公司 2018-06-08 CN disclosed