SCHEMBL28219983

SCHEMBL28219983

Oc1c(Cl)c(Br)nc2cccc(Cl)c12

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
RXFP1 Q9HBX9 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GRIN1 Q05586 4/20 0.40
GRIN2A Q12879 4/20 0.40
ACHE P22303 4/20 0.40
ELANE P08246 2/20 0.39
PARP1 P09874 2/20 0.39
BCHE P06276 2/20 0.39
NQO2 P16083 1/20 0.35
NPC1 O15118 2/20 0.35
DHODH Q02127 1/20 0.35
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28219966 0.83 PARP1 (0.42) GRIN1GRIN2AACHEELANEPARP1
SCHEMBL4787075 0.79 PARP1 (0.46) TSHRMEN1KMT2ARXFP1KDM4E
SCHEMBL626362 0.75 DYRK1A (0.49) TSHRMEN1KMT2ARXFP1KDM4E
Water SCHEMBL25347465 0.73 DYRK1A (0.48) TSHRMEN1KMT2ARXFP1KDM4E
SCHEMBL28219987 0.71 KDM4E (0.42) TSHRKDM4EALDH1A1GRIN1GRIN2A
SCHEMBL18283409 0.70 TDP1 (0.41) GRIN1GRIN2AACHEELANEPARP1
SCHEMBL26607337 0.69 PARP1 (0.43) GRIN1GRIN2AACHEELANEPARP1
SCHEMBL6678089 0.68 PARP1 (0.44) TSHRMEN1KMT2ARXFP1KDM4E
SCHEMBL29344541 0.68 PARP1 (0.42) TSHRMEN1KMT2ARXFP1KDM4E
SCHEMBL28292981 0.68 PARP1 (0.42) GRIN1GRIN2AACHEELANEPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137547-A It can be used as the heterocyclic compound of TNF α conditioning agent 百时美施贵宝公司 2018-06-08 CN disclosed