SCHEMBL28220016

SCHEMBL28220016

Cn1nccc1Cc1cccc(S(C)(=O)=O)c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.40
DRD2 P14416 4/20 0.39
SSTR1 P30872 3/20 0.38
SSTR4 P31391 3/20 0.38
SSTR3 P32745 2/20 0.38
NR1H2 P55055 2/20 0.38
NR1H3 Q13133 1/20 0.38
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CCR1 P32246 1/20 0.36
MET P08581 1/20 0.36
GPR52 Q9Y2T5 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7757122 0.74 KDM5A (0.43) KCNH2ALDH1A1GPR52
SCHEMBL27539141 0.74 KDM4C (0.52)
SCHEMBL17737834 0.70 KMT2A (0.46) NR1H2NR1H3ALDH1A1GAAHSD17B10
SCHEMBL27160505 0.70 RECQL (0.44) DRD2NR1H2NR1H3CYP4F2CYP4A11
SCHEMBL30046411 0.70 HTT (0.56) KCNH2DRD2GAAHSD17B10
SCHEMBL1887800 0.69 TAAR1 (0.46) DRD2NR1H2NR1H3ALDH1A1GAA
SCHEMBL8233359 0.69 ALDH1A1 (0.47) DRD2ALDH1A1GAAHSD17B10SIGMAR1
SCHEMBL7054313 0.69 ALDH1A1 (0.47) DRD2CYP4F2CYP4A11ALDH1A1GAA
SCHEMBL2378354 0.68 ALDH1A1 (0.44) DRD2CYP4F2CYP4A11ALDH1A1GAA
SCHEMBL8278304 0.68 ALDH1A1 (0.51) DRD2ALDH1A1GAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137600-A Condensed pyrazole derivatives as kinase inhibitor UCB生物制药私人有限公司 2018-06-08 CN disclosed