SCHEMBL28220138

SCHEMBL28220138

Nc1[c]cc(C(F)(F)F)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
PLAU P00749 1/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PDE2A O00408 1/20 0.34
GABRA2 P47869 5/20 0.34
GABRB2 P47870 5/20 0.34
GABRP O00591 4/20 0.34
GABRD O14764 4/20 0.34
GABRA1 P14867 4/20 0.34
GABRB1 P18505 4/20 0.34
GABRG2 P18507 4/20 0.34
GABRB3 P28472 4/20 0.34
GABRA5 P31644 4/20 0.34
GABRA3 P34903 4/20 0.34
GABRA4 P48169 4/20 0.34
GABRE P78334 4/20 0.34
GABRA6 Q16445 4/20 0.34
GABRG1 Q8N1C3 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28001125 0.78 TSHR (0.35) POLBTSHRMAPK1GAAGLA
SCHEMBL2333762 0.78 PLAU (0.37) ALDH1A1PLAUKDM4EPOLBSMN1; SMN2
SCHEMBL17238705 0.77 PLAU (0.36) ALDH1A1PLAUKDM4EPOLBSMN1; SMN2
SCHEMBL715069 0.77 PLAU (0.36) ALDH1A1PLAUKDM4EPOLBSMN1; SMN2
SCHEMBL28363679 0.77 TSHR (0.34) PDE2ATSHRMAPK1NOS3NOS2
SCHEMBL630411 0.75 PLAU (0.35) ALDH1A1PLAUKDM4EPOLBSMN1; SMN2
SCHEMBL19471036 0.75 NOTUM (0.35) ALDH1A1PLAUKDM4EPOLBSMN1; SMN2
SCHEMBL27913900 0.72 TSHR (0.34) POLBTSHRMAPK1CYP1A2CYP2C19
SCHEMBL6381071 0.72
SCHEMBL17238695 0.72 PDE2A (0.36) ALDH1A1PLAUKDM4EPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108003162-B Condensed heterocyclic compouds and its application 华南农业大学 2019-02-05 CN disclosed
CN-108003162-A Condensed heterocyclic compouds and its application 华南农业大学 2018-05-08 CN disclosed