SCHEMBL28223403

SCHEMBL28223403

CCOC(=O)c1ccc(N2C(=O)CCC2C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
HTT P42858 4/20 0.52
HPGD P15428 2/20 0.52
HSP90AA1 P07900 2/20 0.52
CACNA1B Q00975 1/20 0.52
APBA1 Q02410 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
MAPK1 P28482 2/20 0.51
GAA P10253 2/20 0.49
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
P2RX3 P56373 2/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
IDO1 P14902 1/20 0.48
TSHR P16473 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14687147 0.80 CA12 (0.53) ALDH1A1HPGDTDP1GAAMEN1
SCHEMBL3003045 0.80 ALDH1A1 (0.48) ALDH1A1HTTHPGDHSP90AA1CACNA1B
SCHEMBL4644173 0.78 ALDH1A1 (0.43) ALDH1A1HPGDTDP1MEN1KMT2A
SCHEMBL11381594 0.77 HTT (0.59) ALDH1A1HTTHPGDHSP90AA1CACNA1B
SCHEMBL16479353 0.76 HTT (0.55) ALDH1A1HTTHPGDHSP90AA1CACNA1B
SCHEMBL16480487 0.76 HDAC2 (0.46) HTTHPGDMAPK1MEN1KMT2A
SCHEMBL4636834 0.76 GAA (0.46) GAAMEN1KMT2ALMNAPOLB
SCHEMBL11112763 0.75 ESR1 (0.49) HSP90AA1NPSR1TDP1MAPK1KMT2A
SCHEMBL7431121 0.74 HTT (0.57) ALDH1A1HTTHPGDHSP90AA1CACNA1B
SCHEMBL9893011 0.74 PER2 (0.40) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108129372-A A kind of method for preparing cyclic lactam derivative 中国科学院大连化学物理研究所 2018-06-08 CN disclosed