SCHEMBL2822378

SCHEMBL2822378

O=C(O)NCCc1cccc(NC(=O)Nc2ccccc2-c2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
NPC1 O15118 1/20 0.51
MAPT P10636 1/20 0.51
RAB9A P51151 1/20 0.51
ITGB1 P05556 2/20 0.47
ITGA4 P13612 2/20 0.47
CA12 O43570 3/20 0.47
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA9 Q16790 3/20 0.47
IDH2 P48735 1/20 0.47
MGLL Q99685 1/20 0.47
GOT1 P17174 1/20 0.47
DDX3X O00571 1/20 0.46
ALDH1A1 P00352 2/20 0.44
TRPV1 Q8NER1 1/20 0.44
LMNA P02545 2/20 0.44
GAA P10253 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2849248 0.86 MEN1 (0.62) MEN1KMT2ANPC1MAPTRAB9A
SCHEMBL1204699 0.85 CA12 (0.52) ITGB1ITGA4CA12CA1CA2
SCHEMBL2823639 0.85 CNR1 (0.57) MEN1KMT2ANPC1MAPTRAB9A
SCHEMBL2827311 0.82 KMT2A (0.72) MEN1KMT2ANPC1MAPTRAB9A
SCHEMBL2824601 0.80 NPC1 (0.61) MEN1KMT2ANPC1MAPTRAB9A
SCHEMBL1205491 0.80 NPSR1 (0.53) MEN1KMT2AMAPTCA12CA1
SCHEMBL2823741 0.79 NPSR1 (0.50) MEN1KMT2ANPC1MAPTRAB9A
SCHEMBL8059186 0.79 KMT2A (0.55) MEN1KMT2ANPC1MAPTRAB9A
SCHEMBL2828371 0.78 MEN1 (0.53) MEN1KMT2ANPC1MAPTRAB9A
SCHEMBL2827217 0.78 HTT (0.56) MEN1KMT2ANPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254860-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR Almirall, S.A. (ES) 2010-12-01 EP disclosed
WO-2009106351-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR ALMIRALL, S.A. (ES) 2009-09-03 WO disclosed
EP-2096105-A1 Derivatives of 4-(2-amino-1-hydroxyethyl)phenol as agonists of the b2 adrenergic receptor Laboratorios Almirall, S.A. (ES) 2009-09-02 EP disclosed