SCHEMBL2849248

SCHEMBL2849248

O=C(O)NCCc1cccc(NC(=O)Nc2ccccc2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.62
KMT2A Q03164 5/20 0.62
NPC1 O15118 3/20 0.62
RAB9A P51151 3/20 0.62
MAPT P10636 3/20 0.62
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
EPHX1 P07099 3/20 0.55
KDM4E B2RXH2 1/20 0.55
CNR1 P21554 5/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
HTR1A P08908 1/20 0.54
DRD2 P14416 1/20 0.54
BTK Q06187 1/20 0.53
LMNA P02545 3/20 0.52
HTT P42858 3/20 0.52
TP53 P04637 2/20 0.52
ALDH1A1 P00352 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2823639 0.93 CNR1 (0.57) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL2827311 0.93 KMT2A (0.72) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL2824601 0.90 NPC1 (0.61) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL8059186 0.89 KMT2A (0.55) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL2827217 0.88 HTT (0.56) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL2850207 0.88 EPHX1 (0.72) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL2826530 0.87 FPR2 (0.65) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL2826334 0.86 KMT2A (0.75) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL2822378 0.86 MEN1 (0.51) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL2828371 0.85 MEN1 (0.53) MEN1KMT2ANPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254860-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR Almirall, S.A. (ES) 2010-12-01 EP disclosed
WO-2009106351-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR ALMIRALL, S.A. (ES) 2009-09-03 WO disclosed
EP-2096105-A1 Derivatives of 4-(2-amino-1-hydroxyethyl)phenol as agonists of the b2 adrenergic receptor Laboratorios Almirall, S.A. (ES) 2009-09-02 EP disclosed