SCHEMBL2824601

SCHEMBL2824601

O=C(O)NCCc1cccc(NC(=O)NCc2ccccc2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.61
RAB9A P51151 5/20 0.61
MEN1 O00255 4/20 0.61
KMT2A Q03164 4/20 0.61
MAPT P10636 2/20 0.61
EPHX1 P07099 2/20 0.59
SMN1; SMN2 Q16637 5/20 0.57
TP53 P04637 2/20 0.57
HPGD P15428 1/20 0.57
KDR P35968 1/20 0.56
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
HTT P42858 2/20 0.54
POLB P06746 1/20 0.54
MAOB P27338 1/20 0.54
NAMPT P43490 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.52
GSK3B P49841 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2827311 0.92 KMT2A (0.72) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL2853369 0.91 RAB9A (0.65) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL2849248 0.90 MEN1 (0.62) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL2823977 0.88 RAB9A (0.54) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL2823579 0.87 KMT2A (0.60) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL2850207 0.86 EPHX1 (0.72) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL2826334 0.85 KMT2A (0.75) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL8059186 0.85 KMT2A (0.55) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL1206039 0.84 KDR (0.57) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL2823639 0.84 CNR1 (0.57) NPC1RAB9AMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101939291-A Derivatives of 4-(2-amino-1-hydroxyethyl)phenol as agonists of the beta2 adrenergic receptor AMIRALL S A 2011-01-05 CN disclosed
EP-2254860-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR Almirall, S.A. (ES) 2010-12-01 EP disclosed
WO-2009106351-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR ALMIRALL, S.A. (ES) 2009-09-03 WO disclosed
EP-2096105-A1 Derivatives of 4-(2-amino-1-hydroxyethyl)phenol as agonists of the b2 adrenergic receptor Laboratorios Almirall, S.A. (ES) 2009-09-02 EP disclosed