Pyridazine

Pyridazine

SCHEMBL28223809

CC(C)OC(=O)NN.c1ccnnc1

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.36
ALOX15 P16050 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
RAB9A P51151 1/20 0.35
HTT P42858 1/20 0.35
P2RX7 Q99572 2/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
TSHR P16473 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAP3K5 Q99683 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1134094 0.83
Furan SCHEMBL27965211 0.77 HPGD (0.36) HPGDALOX15SMN1; SMN2NPC1CYP1A2
Pyridazine SCHEMBL27835452 0.73 APLNR (0.38) NPC1RAB9AP2RX7CA12CA1
Pyridazine SCHEMBL27711578 0.69 P2RX7 (0.43) SMN1; SMN2CYP1A2CYP2D6CYP2C9CYP2C19
Pyridazine SCHEMBL27723556 0.68 SMN1; SMN2 (0.35) SMN1; SMN2CA12CA14ALDH1A1
SCHEMBL28257017 0.68 KDM4E (0.39) SMN1; SMN2HDAC1HDAC2TSHRKDM4E
SCHEMBL11428405 0.68
SCHEMBL13738164 0.68
SCHEMBL441968 0.65 TSHR (0.46) HPGDALOX15SMN1; SMN2NPC1CYP1A2
SCHEMBL10592352 0.64 HCAR2 (0.53) CYP2C9HTTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088101-A A kind of nitrogen-containing hetero cyclics, preparation method, pharmaceutical composition and application 罗欣药业(上海)有限公司 2019-08-02 CN disclosed
CN-108069959-A A kind of nitrogen-containing hetero cyclics, its preparation method, pharmaceutical composition and application 凯惠科技发展(上海)有限公司 2018-05-25 CN disclosed