SCHEMBL2822644

SCHEMBL2822644

O=C(CCc1ccc(OCc2ccc(CN3CCCC3c3ccccc3)cc2)cc1)OC(=O)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.48
OPRK1 P41145 1/20 0.48
HRH3 Q9Y5N1 9/20 0.46
SPHK1 Q9NYA1 4/20 0.44
SPHK2 Q9NRA0 3/20 0.44
SCN3A Q9NY46 1/20 0.43
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
LTA4H P09960 2/20 0.42
EPHX2 P34913 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
FFAR1 O14842 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2822642 0.89 FFAR1 (0.53) OPRM1OPRK1HRH3SPHK1SPHK2
SCHEMBL2824720 0.89 HRH3 (0.42) HRH3SPHK1SPHK2SCN3AMAOA
SCHEMBL2824092 0.87 SPHK1 (0.52) HRH3SPHK1SPHK2MAOAMAOB
SCHEMBL2826434 0.87 SPHK1 (0.52) HRH3SPHK1SPHK2MAOAMAOB
SCHEMBL13887158 0.86 FFAR1 (0.58) OPRM1OPRK1HRH3SPHK1SPHK2
SCHEMBL2827661 0.84 HRH3 (0.42) HRH3SPHK1SPHK2SCN3AMAOA
SCHEMBL2827471 0.84 HRH3 (0.44) HRH3SPHK1SCN3AMAOAMAOB
SCHEMBL2827613 0.83 LTA4H (0.53) HRH3LTA4HEPHX2NPC1RAB9A
Trifluoroacetic Acid SCHEMBL2824716 0.79 FFAR1 (0.49) HRH3SPHK1FFAR1FFAR4
SCHEMBL2823889 0.78 LTA4H (0.65) HRH3LTA4HEPHX2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1731505-B1 ALKOXYPHENYLPROPANOIC ACID DERIVATIVES TAKEDA PHARMACEUTICAL (JP) 2015-01-14 EP disclosed
EP-2253315-A1 Alkoxyphenylpropanoic acid derivatives Takeda Pharmaceutical Company Limited (JP) 2010-11-24 EP disclosed
EP-1731505-A1 ALKOXYPHENYLPROPANOIC ACID DERIVATIVES Takeda Pharmaceutical Company Limited (JP) 2006-12-13 EP disclosed