SCHEMBL28243763

SCHEMBL28243763

Cc1ccnc(I)c1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.38
ALDH1A1 P00352 4/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
LMNA P02545 1/20 0.36
NAPRT Q6XQN6 1/20 0.36
P4HTM Q9NXG6 1/20 0.36
ASPH Q12797 2/20 0.36
KDM8 Q8N371 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
SIRT3 Q9NTG7 1/20 0.36
MAPK1 P28482 1/20 0.36
NOTUM Q6P988 1/20 0.35
KDM5A P29375 2/20 0.35
KDM4C Q9H3R0 2/20 0.35
KDM5B Q9UGL1 2/20 0.35
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
KDM6B O15054 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17611245 0.80 NAPRT (0.46) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL28280472 0.79 KDM4E (0.38) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL353204 0.79 KDM4E (0.40) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL10766873 0.78 CYP3A4 (0.39) KDM4EALDH1A1L3MBTL1TDP1LMNA
Hydrochloric Acid SCHEMBL4249059 0.78 KDM4E (0.39) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL9684174 0.78 KDM4E (0.50) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL7612137 0.78 L3MBTL1 (0.38) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL9504653 0.78 KDM4E (0.39) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL30049082 0.78 KDM4E (0.50) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL8895032 0.77 ALDH1A1 (0.36) KDM4EALDH1A1L3MBTL1ASPHKDM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104341425-B Deuterated acetylene-derivative, its pharmaceutical composition and application 上海医药集团股份有限公司 2018-11-02 CN disclosed