SCHEMBL28248171

SCHEMBL28248171

c1cnc(NC2(c3cccnc3)CCC2)nc1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 9/20 0.58
HDAC6 Q9UBN7 11/20 0.51
HDAC3 O15379 10/20 0.48
HDAC1 Q13547 10/20 0.48
HDAC2 Q92769 10/20 0.48
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
BTD P43251 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24967744 0.88 VNN1 (0.56) VNN1HDAC6HDAC3HDAC1HDAC2
SCHEMBL28247582 0.83 HDAC6 (0.60) VNN1HDAC6HDAC3HDAC1HDAC2
SCHEMBL18742418 0.80 VNN1 (0.64) VNN1HDAC6HDAC3HDAC1HDAC2
SCHEMBL28248162 0.80 HDAC6 (0.60) VNN1HDAC6HDAC3HDAC1HDAC2
SCHEMBL28248331 0.78 HDAC6 (0.61) VNN1HDAC6HDAC3HDAC1HDAC2
SCHEMBL18742570 0.77 VNN1 (0.59) VNN1HDAC6HDAC3HDAC1HDAC2
SCHEMBL28247580 0.75 HDAC6 (0.49) VNN1HDAC6HDAC3HDAC1HDAC2
SCHEMBL28248252 0.75 HDAC6 (0.52) VNN1HDAC6HDAC3HDAC1HDAC2
SCHEMBL28247670 0.75 HDAC6 (0.57) VNN1HDAC6HDAC3HDAC1HDAC2
SCHEMBL18742532 0.75 HDAC6 (0.92) HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108699048-A Oxadiazolamide derivative compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions comprising the same 株式会社钟根堂 2018-10-23 CN disclosed