SCHEMBL28249003

SCHEMBL28249003

C1=CC=CNC=C1.O=C(O)C1Cc2cccc3cccc1c23

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 9/20 0.42
MTNR1B P49286 9/20 0.42
ALDH1A1 P00352 1/20 0.38
KDM4E B2RXH2 1/20 0.37
OPRL1 P41146 7/20 0.36
OPRM1 P35372 6/20 0.36
OPRK1 P41145 5/20 0.36
OPRD1 P41143 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30066901 0.88 MTNR1A (0.50) MTNR1AMTNR1BALDH1A1KDM4EOPRL1
SCHEMBL5380872 0.88 MTNR1A (0.50) MTNR1AMTNR1BALDH1A1KDM4EOPRL1
SCHEMBL28248972 0.88 MTNR1A (0.41) MTNR1AMTNR1BKDM4EOPRL1OPRM1
Hydrochloric Acid SCHEMBL28260890 0.86 MTNR1A (0.40) MTNR1AMTNR1BKDM4EOPRL1OPRM1
SCHEMBL28249001 0.84 MTNR1A (0.44) MTNR1AMTNR1BOPRL1OPRM1
SCHEMBL9240061 0.77 MTNR1A (0.51) MTNR1AMTNR1BKDM4EOPRL1OPRM1
SCHEMBL28249002 0.76 MTNR1A (0.38) MTNR1AMTNR1BKDM4EOPRL1OPRM1
SCHEMBL28260913 0.75 MTNR1A (0.37) MTNR1AMTNR1BKDM4EOPRL1OPRM1
SCHEMBL11146721 0.75 MTNR1A (0.47) MTNR1AMTNR1BKDM4EOPRL1OPRM1
SCHEMBL5370015 0.74 MTNR1A (0.56) MTNR1AMTNR1BKDM4EOPRL1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071563-A Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2018-12-21 CN claimed
CN-109071563-A Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2018-12-21 CN disclosed
CN-108884106-A POLYCYCLIC COMPOUNDS AS INHIBITORS OF BRUTON'S TYROSINE KINASE 詹森药业有限公司 2018-11-23 CN disclosed