SCHEMBL28249233

SCHEMBL28249233

CC(C)CCN1CCC(NC(=O)OC(C)(C)C)C1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.54
HRH2 P25021 4/20 0.49
HRH1 P35367 4/20 0.49
CCR5 P51681 1/20 0.49
KCNA3 P22001 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
HSD11B1 P28845 5/20 0.46
CYP2C9 P11712 1/20 0.46
DRD2 P14416 2/20 0.42
BTK Q06187 1/20 0.42
JAK2 O60674 2/20 0.41
JAK1 P23458 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011587 0.93 CCR5 (0.55) CTSKHRH2HRH1CCR5KCNA3
SCHEMBL25326818 0.92 CA1 (0.54) CTSKHRH2HRH1CCR5KCNA3
SCHEMBL10280626 0.86 CTSK (0.57) CTSKHRH2HRH1CCR5KCNA3
SCHEMBL18530346 0.86 CTSK (0.57) CTSKHRH2HRH1CCR5KCNA3
SCHEMBL13102176 0.86 CTSK (0.57) CTSKHRH2HRH1CCR5KCNA3
SCHEMBL13583572 0.86 CTSK (0.57) CTSKHRH2HRH1CCR5KCNA3
SCHEMBL13583571 0.86 CTSK (0.57) CTSKHRH2HRH1CCR5KCNA3
SCHEMBL13102166 0.86 CTSK (0.57) CTSKHRH2HRH1CCR5KCNA3
SCHEMBL1810659 0.85 CTSK (0.56) CTSKHRH2HRH1CCR5KCNA3
SCHEMBL1700413 0.85 CTSK (0.56) CTSKHRH2HRH1CCR5KCNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727343-A Quinazolinones PARP-1/2 inhibitor containing 3- amino nafoxidines and preparation method thereof, pharmaceutical composition and purposes 中国医学科学院药物研究所 2018-11-02 CN disclosed