SCHEMBL28250100

SCHEMBL28250100

COC(=O)C[C@H](Nc1ccccc1)C(=O)OC

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.48
CA2 P00918 2/20 0.48
CA9 Q16790 2/20 0.48
CA1 P00915 1/20 0.48
KMT2A Q03164 2/20 0.46
ATM Q13315 1/20 0.42
ALDH1A1 P00352 2/20 0.41
THRB P10828 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41
POLB P06746 2/20 0.40
KCNA5 P22460 1/20 0.40
LMNA P02545 1/20 0.40
ABCB1 P08183 1/20 0.39
GAA P10253 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13660425 1.00 CA12 (0.48) CA12CA2CA9CA1KMT2A
SCHEMBL7028330 0.91 CA12 (0.43) CA12CA2CA9CA1KMT2A
SCHEMBL27257857 0.86 KLK5 (0.45) CA12CA2CA9CA1KMT2A
SCHEMBL13881222 0.86 ITGA4 (0.45) CA12CA2CA9CA1KMT2A
SCHEMBL5930583 0.84 CA12 (0.43) CA12CA2CA9CA1ALDH1A1
SCHEMBL11481798 0.83 CA12 (0.49) CA12CA2CA9CA1KMT2A
SCHEMBL6951139 0.83 ALDH1A1 (0.50) CA12CA2CA9CA1KMT2A
SCHEMBL6951142 0.83 ALDH1A1 (0.50) CA12CA2CA9CA1KMT2A
SCHEMBL5936826 0.83 KMT2A (0.47) CA12CA2CA9KMT2AATM
SCHEMBL22661871 0.83 KMT2A (0.47) CA12CA2CA9KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105392788-B Substituted bridging urea analog as Sirtuin conditioning agent 葛兰素史密斯克莱有限责任公司 2018-10-23 CN disclosed