SCHEMBL28255102

SCHEMBL28255102

COC1(c2ccccc2)CCCC1.O=S(=O)(Cl)Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.50
OPRM1 P35372 2/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
OPRL1 P41146 1/20 0.47
ALOX5 P09917 1/20 0.41
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
DRD3 P35462 1/20 0.39
GAA P10253 1/20 0.39
MCOLN3 Q8TDD5 1/20 0.39
AKR1C1 Q04828 1/20 0.39
SCD5 Q86SK9 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14899046 0.89 OPRM1 (0.56) HSD11B1OPRM1OPRD1OPRK1OPRL1
SCHEMBL1040389 0.87 OPRM1 (0.54) HSD11B1OPRM1OPRD1OPRK1OPRL1
SCHEMBL16024156 0.87 OPRM1 (0.54) HSD11B1OPRM1OPRD1OPRK1OPRL1
SCHEMBL1040539 0.87 OPRM1 (0.54) HSD11B1OPRM1OPRD1OPRK1OPRL1
SCHEMBL10821867 0.85 OPRM1 (0.56) HSD11B1OPRM1OPRD1OPRK1OPRL1
SCHEMBL19126917 0.81 HSD11B1 (0.43) HSD11B1OPRM1OPRD1OPRK1OPRL1
SCHEMBL13876257 0.80 OPRM1 (0.59) HSD11B1OPRM1OPRD1OPRK1OPRL1
SCHEMBL778919 0.76 GAA (0.42) HSD11B1PSEN1PSEN2APH1BNCSTN
SCHEMBL776247 0.74 PSEN1 (0.42) OPRM1OPRD1PSEN1PSEN2APH1B
SCHEMBL6132219 0.74 MEN1 (0.57) HSD11B1OPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884093-A 6,7,8,9- tetrahydro -5H- pyrido [2,3-d] azepine * dopamine D 3 ligands 辉瑞公司 2018-11-23 CN disclosed