SCHEMBL28255683

SCHEMBL28255683

O=C1Nc2cccc(N3CCCC3)c2C1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.53
ALDH1A1 P00352 3/20 0.53
MAPK1 P28482 3/20 0.53
L3MBTL1 Q9Y468 3/20 0.53
EGFR P00533 2/20 0.53
RAF1 P04049 1/20 0.53
ALOX12 P18054 1/20 0.53
MAP2K1 Q02750 1/20 0.53
CES1 P23141 2/20 0.50
NSD2 O96028 1/20 0.48
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
EEF2K O00418 1/20 0.42
ERBB2 P04626 1/20 0.39
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
KDM4E B2RXH2 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
GAA P10253 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6888226 0.87 CES1 (0.47) ALDH1A1CES1KDM4ELMNA
SCHEMBL4202385 0.79 MAPT (0.63) MAPTALDH1A1L3MBTL1TDP1NPSR1
SCHEMBL13244107 0.76 BACE1 (0.46) MAPTALDH1A1MAPK1LMNA
SCHEMBL28522247 0.73 MAPT (0.57) MAPTALDH1A1MAPK1L3MBTL1EGFR
Hydrochloric Acid SCHEMBL15282882 0.72 MAPT (0.55) MAPTALDH1A1MAPK1L3MBTL1EGFR
SCHEMBL2463193 0.69 MAPT (1.00) MAPTALDH1A1MAPK1L3MBTL1EGFR
SCHEMBL28339971 0.68 MAPT (0.54) MAPTALDH1A1MAPK1L3MBTL1EGFR
SCHEMBL3273424 0.68 MAPT (0.97) MAPTALDH1A1MAPK1L3MBTL1EGFR
Isatin SCHEMBL4625841 0.68 MAOA (0.69) ALDH1A1MAOAMAOBERBB2KMT2A
SCHEMBL4242823 0.67 CES1 (0.60) MAPTCES1MAOAMAOBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108912127-B Benzo [ b, e ] azepine compound based on isatin skeleton and preparation method thereof 青岛农业大学 2019-12-10 CN claimed
CN-108912127-A A kind of benzo [b, e] azatropylidene compound and preparation method thereof based on isatin skeleton 青岛农业大学 2018-11-30 CN claimed
CN-112574108-B Preparation method of polysubstituted benzo [ b ] azepine compound 甘肃兴荣精细化工有限公司 2023-08-11 CN disclosed
CN-112574108-A Preparation method of polysubstituted benzo [ b ] aza compound 兰州大学 2021-03-30 CN disclosed
CN-108912127-B Benzo [ b, e ] azepine compound based on isatin skeleton and preparation method thereof 青岛农业大学 2019-12-10 CN disclosed
CN-108912127-B Benzo [ b, e ] azepine compound based on isatin skeleton and preparation method thereof 青岛农业大学 2019-12-10 CN disclosed
CN-108912127-A A kind of benzo [b, e] azatropylidene compound and preparation method thereof based on isatin skeleton 青岛农业大学 2018-11-30 CN disclosed
CN-108912127-A A kind of benzo [b, e] azatropylidene compound and preparation method thereof based on isatin skeleton 青岛农业大学 2018-11-30 CN disclosed