SCHEMBL28256752

SCHEMBL28256752

COC(=O)/C(=C/c1ccccc1OCc1ccccc1)CC(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 1/20 0.52
CDK1 P06493 1/20 0.52
CDK4 P11802 1/20 0.52
CCNB1 P14635 1/20 0.52
CCND1 P24385 1/20 0.52
CCNB3 Q8WWL7 1/20 0.52
PTGER1 P34995 1/20 0.51
PTGER4 P35408 1/20 0.51
PTGER3 P43115 1/20 0.51
PTGER2 P43116 1/20 0.51
KDM4E B2RXH2 4/20 0.48
LMNA P02545 3/20 0.48
ALDH1A1 P00352 3/20 0.48
HPGD P15428 2/20 0.48
RECQL P46063 1/20 0.48
BRD4 O60885 1/20 0.47
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
POLB P06746 1/20 0.45
PKM P14618 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3959188 1.00 CCNB2 (0.52) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL3959185 0.79 NR1H4 (0.60) KDM4EALDH1A1RECQLKMT2AMEN1
SCHEMBL17318680 0.77 RECQL (0.45) LMNAALDH1A1RECQLKMT2AMEN1
SCHEMBL17318679 0.77 RECQL (0.45) LMNAALDH1A1RECQLKMT2AMEN1
SCHEMBL17318678 0.77 RECQL (0.45) LMNAALDH1A1RECQLKMT2AMEN1
SCHEMBL27252480 0.77 CCNB2 (0.47) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL16303657 0.77 CCNB2 (0.47) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL3960454 0.76 LMNA (0.46) PTGER1PTGER4PTGER3PTGER2LMNA
SCHEMBL3967797 0.76 KDM4E (0.56) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL3520152 0.76 LMNA (0.46) PTGER1PTGER4PTGER3PTGER2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115385886-B AcrB efflux pump inhibitor and preparation method and application thereof 山东大学 2024-04-19 CN disclosed
CN-108822095-B Benzo [ h ] chromene compound and application thereof as AcrB efflux pump inhibitor in antibiosis 山东大学 2020-05-01 CN disclosed
CN-108822095-A Benzo [h] chromene compound and its application as AcrB efflux pump inhibitor in antibacterial 山东大学 2018-11-16 CN disclosed