SCHEMBL28258378

SCHEMBL28258378

CCN(CC)C(=O)C1CCCN(c2ccccc2)C1

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.70
MAPT P10636 2/20 0.70
MAPK1 P28482 1/20 0.70
KDM4E B2RXH2 3/20 0.65
LMNA P02545 1/20 0.64
HPGD P15428 1/20 0.61
HSD17B10 Q99714 1/20 0.58
POLB P06746 1/20 0.55
GAA P10253 1/20 0.55
NOTUM Q6P988 1/20 0.52
BCL9 O00512 1/20 0.52
CTNNB1 P35222 1/20 0.52
TP53 P04637 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
HTT P42858 1/20 0.52
CTSB P07858 1/20 0.52
ACACB O00763 1/20 0.50
ACACA Q13085 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12006548 0.87 ALDH1A1 (0.71) ALDH1A1MAPTMAPK1KDM4ELMNA
SCHEMBL3455666 0.83 ALDH1A1 (1.00) ALDH1A1MAPTMAPK1KDM4ELMNA
SCHEMBL4961935 0.79 NOTUM (0.81) ALDH1A1MAPTMAPK1KDM4EHSD17B10
SCHEMBL613112 0.79 NOTUM (0.81) ALDH1A1MAPTMAPK1KDM4EHSD17B10
SCHEMBL14504051 0.79 ALDH1A1 (0.61) ALDH1A1MAPTMAPK1KDM4ELMNA
SCHEMBL3455456 0.78 ALDH1A1 (1.00) ALDH1A1MAPTMAPK1KDM4ELMNA
SCHEMBL31175186 0.78 ALDH1A1 (0.70) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL12777820 0.78 KDM4E (0.60) ALDH1A1MAPTKDM4ELMNAHPGD
SCHEMBL12311912 0.78 ALDH1A1 (0.59) ALDH1A1MAPTMAPK1KDM4ELMNA
SCHEMBL2446475 0.77 KMT2A (0.62) ALDH1A1MAPTMAPK1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715617-A Dimethoxyphenyl-substituted indole compounds as inhibitors of TLR7, TLR8 or TLR9 百时美施贵宝公司 2019-05-03 CN claimed
CN-109715617-A Dimethoxyphenyl-substituted indole compounds as inhibitors of TLR7, TLR8 or TLR9 百时美施贵宝公司 2019-05-03 CN disclosed
CN-109641895-A Indole compounds substituted with [1, 2, 4] triazolo [1, 5-a ] pyridyl 百时美施贵宝公司 2019-04-16 CN disclosed
CN-104876955-B Arginase inhibitor and its treatment use 马尔斯公司 2018-11-23 CN disclosed