SCHEMBL28258656

SCHEMBL28258656

NC(=O)c1ccc2c(C(N)=O)n[nH]c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.53
JAK2 O60674 1/20 0.52
JAK1 P23458 1/20 0.52
TYK2 P29597 1/20 0.52
JAK3 P52333 1/20 0.52
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47
MAP2K4 P45985 7/20 0.47
MAPK1 P28482 2/20 0.47
MAPK6 Q16659 2/20 0.47
MAPKAPK2 P49137 1/20 0.47
MAPKAPK3 Q16644 1/20 0.47
MAPKAPK5 Q8IW41 1/20 0.47
AAK1 Q2M2I8 2/20 0.46
PARP1 P09874 1/20 0.43
CHEK2 O96017 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK10 P53779 1/20 0.41
MAPK14 Q16539 1/20 0.41
CDK7 P50613 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13386744 0.90 JAK2 (0.50) CHEK1JAK2JAK1TYK2JAK3
SCHEMBL31033009 0.86 CHEK1 (0.53) CHEK1JAK2JAK1MAP2K4MAPK1
SCHEMBL19773425 0.84 CHEK1 (0.52) CHEK1JAK2JAK1TYK2JAK3
SCHEMBL8877902 0.84 JAK1 (0.65) CHEK1JAK2JAK1TYK2JAK3
SCHEMBL19208914 0.83 JAK2 (0.59) CHEK1JAK2JAK1TYK2JAK3
SCHEMBL16252829 0.83 MAP2K4 (0.52) JAK2JAK1TYK2JAK3MAP2K4
SCHEMBL31173858 0.83 MAP2K4 (0.51) CHEK1JAK2JAK1TYK2JAK3
SCHEMBL15540985 0.83 MAP2K4 (0.52) CHEK1JAK2JAK1TYK2JAK3
SCHEMBL5051796 0.83 CHEK1 (0.54) CHEK1MAP2K4MAPK1MAPK6MAPKAPK2
SCHEMBL15541582 0.83 JAK2 (0.53) JAK2JAK1TYK2JAK3ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109121414-A Benzopyrazole compounds and analogs thereof 拜奥克里斯特制药公司 2019-01-01 CN disclosed