SCHEMBL28259792

SCHEMBL28259792

O=C(O)c1scc(Br)c1[N+](=O)[O-]

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 8/20 0.41
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GSK3B P49841 2/20 0.36
ESR2 Q92731 1/20 0.36
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
RAB9A P51151 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23485282 0.81 GPR35 (0.36) GPR35ALDH1A1L3MBTL1ESR2TDP1
SCHEMBL11481751 0.79 TDP1 (0.46) GPR35ALDH1A1L3MBTL1ESR2TSHR
SCHEMBL28866506 0.79 COMT (0.46) ALDH1A1L3MBTL1TSHRCYP1A2CYP2C19
SCHEMBL16737142 0.76 ESR2 (0.41) GPR35ALDH1A1L3MBTL1GSK3BESR2
SCHEMBL4584130 0.70 GSK3B (0.59) GPR35L3MBTL1GSK3BTSHRTDP1
SCHEMBL3281960 0.69 GPR35 (0.47) GPR35L3MBTL1GSK3BTSHRTDP1
SCHEMBL1973884 0.69 GPR35 (0.47) GPR35L3MBTL1GSK3BTSHRTDP1
SCHEMBL1475958 0.68 CA1 (0.42) GPR35ALDH1A1L3MBTL1TSHRTDP1
SCHEMBL6593908 0.68 TSHR (0.46) GPR35ALDH1A1L3MBTL1ESR2TSHR
SCHEMBL16737121 0.68 GPR35 (0.36) GPR35ALDH1A1L3MBTL1GSK3BESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884066-B 2, 3, 5-substituted thiophene compounds as protein kinase inhibitors 韩国科学技术研究院 2021-08-24 CN disclosed
CN-108884066-A The thiophene compound that new 2,3,5- as kinases inhibitor replace 韩国科学技术研究院 2018-11-23 CN disclosed